Assay

PGDB_AS002101

System: biochemicalTarget: CRBN
Assay context summary

Assay context

4 activity records
Assay familybiochemical
Systembiochemical
ReadoutIC50
TargetCRBN
E3CRBN
OrganismHomo sapiens
TechnologyHTRF
Activity compounds and values

Activity records

4 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C020138
IC50-=1.5-1.9uM-—CRBNCRBN-WO2024245444A1PGDB_A028177PGDB_C020138PGDB_AS002101View
2D structure for PGDB_C014239
IC50-=1-1.5uM-—CRBNCRBN-WO2024245444A1PGDB_A040550PGDB_C014239PGDB_AS002101View
2D structure for PGDB_C019997
IC50-=1.5-1.9uM-—CRBNCRBN-WO2024245444A1PGDB_A044235PGDB_C019997PGDB_AS002101View
2D structure for PGDB_C019943
IC50-=1-1.5uM-—CRBNCRBN-WO2024245444A1PGDB_A075089PGDB_C019943PGDB_AS002101View
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