Assay

PGDB_AS002316

System: cell_basedTarget: GSPT1Cell line: 293GT
Assay context summary

Assay context

57 activity records
Assay family% Degradation
Systemcell_based
ReadoutEC50
TargetGSPT1
E3CRBN
Cell line293GT
OrganismHomo sapiens
Technologyluminescence
Detection targetprotein_degradation
Activity compounds and values

Activity records

57 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C022693
EC50->30.0uM-—--293GTCN111051298APGDB_A007341PGDB_C022693PGDB_AS002316View
2D structure for PGDB_C022654
EC50->30.0uM-—--293GTCN111051298APGDB_A007950PGDB_C022654PGDB_AS002316View
2D structure for PGDB_C022773
EC50->30uM-—--293GTCN111051298APGDB_A011076PGDB_C022773PGDB_AS002316View
2D structure for PGDB_C022680
EC50->30.0uM-—--293GTCN111051298APGDB_A013005PGDB_C022680PGDB_AS002316View
2D structure for PGDB_C022774
EC50->30uM-—--293GTCN111051298APGDB_A014003PGDB_C022774PGDB_AS002316View
2D structure for PGDB_C022644
EC50->50.0uM-—--293GTCN111051298APGDB_A014541PGDB_C022644PGDB_AS002316View
2D structure for PGDB_C022769
EC50->50uM-—--293GTCN111051298APGDB_A014694PGDB_C022769PGDB_AS002316View
2D structure for PGDB_C022628
EC50->50.0uM-—--293GTCN111051298APGDB_A014699PGDB_C022628PGDB_AS002316View
2D structure for PGDB_C022637
EC50->50.0uM-—--293GTCN111051298APGDB_A016340PGDB_C022637PGDB_AS002316View
2D structure for PGDB_C022715
EC50->30.0uM-—--293GTCN111051298APGDB_A016464PGDB_C022715PGDB_AS002316View
2D structure for PGDB_C022642
EC50->50.0uM-—--293GTCN111051298APGDB_A018962PGDB_C022642PGDB_AS002316View
2D structure for PGDB_C022652
EC50->30.0uM-—--293GTCN111051298APGDB_A019325PGDB_C022652PGDB_AS002316View
2D structure for PGDB_C022723
EC50->30uM-—--293GTCN111051298APGDB_A020703PGDB_C022723PGDB_AS002316View
2D structure for PGDB_C022658
EC50->30.0uM-—--293GTCN111051298APGDB_A022144PGDB_C022658PGDB_AS002316View
2D structure for PGDB_C022681
EC50->30.0uM-—--293GTCN111051298APGDB_A022365PGDB_C022681PGDB_AS002316View
2D structure for PGDB_C022752
EC50->30uM-—--293GTCN111051298APGDB_A022401PGDB_C022752PGDB_AS002316View
2D structure for PGDB_C022675
EC50->30.0uM-—--293GTCN111051298APGDB_A022607PGDB_C022675PGDB_AS002316View
2D structure for PGDB_C022730
EC50->30.0uM-—--293GTCN111051298APGDB_A022833PGDB_C022730PGDB_AS002316View
2D structure for PGDB_C022653
EC50->30.0uM-—--293GTCN111051298APGDB_A026723PGDB_C022653PGDB_AS002316View
2D structure for PGDB_C022638
EC50->50.0uM-—--293GTCN111051298APGDB_A027123PGDB_C022638PGDB_AS002316View
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