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O=C1CCC(N2Cc3cc(C4CCN(Cc5ccc(-c6ccccc6)cc5)CC4)ccc3C2=O)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | > | 50.0 | uM | - | — | - | - | 293GT | CN111051298A | PGDB_A018962 | PGDB_C022642 | PGDB_AS002316 | View | |
| EC50 | - | > | 50.0 | uM | - | — | - | - | 293GT | CN111051298A | PGDB_A019428 | PGDB_C022642 | PGDB_AS000334 | View | |
| EC50 | - | = | 0.007 | uM | - | — | - | - | 293GT | CN111051298A | PGDB_A023000 | PGDB_C022642 | PGDB_AS001169 | View | |
| EC50 | - | > | 50.0 | uM | - | — | - | - | 293GT | CN111051298A | PGDB_A029542 | PGDB_C022642 | PGDB_AS002316 | View | |
| EC50 | - | > | 50.0 | uM | - | — | - | - | 293GT | CN111051298A | PGDB_A049938 | PGDB_C022642 | PGDB_AS000334 | View | |
| EC50 | - | = | 0.007 | uM | - | — | - | - | 293GT | CN111051298A | PGDB_A052108 | PGDB_C022642 | PGDB_AS001169 | View | |
| % Degradation | - | = | 65.0 | % | 10 uM | 24 h | - | - | 293GT | CN111051298A | PGDB_A054023 | PGDB_C022642 | PGDB_AS002112 | View | |
| % Degradation | - | = | 65.0 | % | 10 uM | 24 h | - | - | 293GT | CN111051298A | PGDB_A056125 | PGDB_C022642 | PGDB_AS002112 | View |