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Compound
PGDB_C002218
6 activity records1 related patents
2D structure
O=C1CCC(N2C(=O)c3cccc(NCc4cccc(NC(=O)[C@H]5CC[C@H](c6nc7cccnc7s6)CC5)c4F)c3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GI50 | - | = | 11.38 | nM | - | — | GSPT1 | - | SU-DHL-2 | WO2023237116A1 | PGDB_A013438 | PGDB_C002218 | PGDB_AS000205 | View |
| GI50 | - | = | 0.33 | nM | - | — | GSPT1 | - | Toledo | WO2023237116A1 | PGDB_A024930 | PGDB_C002218 | PGDB_AS002036 | View |
| GI50 | - | = | 4.03 | nM | - | — | GSPT1 | - | Raji | WO2023237116A1 | PGDB_A036142 | PGDB_C002218 | PGDB_AS000230 | View |
| GI50 | - | < | 100 | nM | - | — | GSPT1 | - | HL-60 | WO2023237116A1 | PGDB_A047435 | PGDB_C002218 | PGDB_AS001555 | View |
| GI50 | - | = | 5.62 | nM | - | — | GSPT1 | - | Hep3B | WO2023237116A1 | PGDB_A062143 | PGDB_C002218 | PGDB_AS001914 | View |
| DC50 | - | < | 100 | nM | - | — | GSPT1 | - | HEK293 | WO2023237116A1 | PGDB_A073056 | PGDB_C002218 | PGDB_AS002200 | View |