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Compound
PGDB_C002259
5 activity records1 related patents
2D structure
Cn1c2cnccc2nc1[C@H]1CC[C@H](N2Cc3ccc(CNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3C2=O)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GI50 | - | = | 22.29 | nM | - | — | GSPT1 | - | Hep3B | WO2023237116A1 | PGDB_A009004 | PGDB_C002259 | PGDB_AS001914 | View |
| GI50 | - | = | 5.21 | nM | - | — | GSPT1 | - | NCI-H929 | WO2023237116A1 | PGDB_A024168 | PGDB_C002259 | PGDB_AS000710 | View |
| GI50 | - | < | 100 | nM | - | — | GSPT1 | - | HL-60 | WO2023237116A1 | PGDB_A039918 | PGDB_C002259 | PGDB_AS001555 | View |
| GI50 | - | = | 1.63 | nM | - | — | GSPT1 | - | Toledo | WO2023237116A1 | PGDB_A040115 | PGDB_C002259 | PGDB_AS002036 | View |
| DC50 | - | < | 100 | nM | - | — | GSPT1 | - | HEK293 | WO2023237116A1 | PGDB_A067290 | PGDB_C002259 | PGDB_AS002200 | View |