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Compound
PGDB_C002262
4 activity records1 related patents
2D structure
COc1ccc(CNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1C(=O)N[C@H]1CC[C@H](c2nc3ccncc3n2C)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GI50 | - | < | 100 | nM | - | — | GSPT1 | - | HL-60 | WO2023237116A1 | PGDB_A033322 | PGDB_C002262 | PGDB_AS001555 | View |
| DC50 | - | < | 100 | nM | - | — | GSPT1 | - | HEK293 | WO2023237116A1 | PGDB_A046650 | PGDB_C002262 | PGDB_AS002200 | View |
| GI50 | - | = | 1.42 | nM | - | — | GSPT1 | - | Hep3B | WO2023237116A1 | PGDB_A051277 | PGDB_C002262 | PGDB_AS001914 | View |
| GI50 | - | = | 0.5 | nM | - | — | GSPT1 | - | SU-DHL-2 | WO2023237116A1 | PGDB_A077636 | PGDB_C002262 | PGDB_AS000205 | View |