Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C003184
4 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(Cn4cc(Cc5cccc(Br)c5)nn4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GI50 | - | = | 4.5 | nM | - | — | GSPT1 | - | NB4 | WO2024222614A1 | PGDB_A014707 | PGDB_C003184 | PGDB_AS001086 | View |
| Dmax | - | = | 113 | % | - | 4 h | GSPT1 | - | NB4 | WO2024222614A1 | PGDB_A015376 | PGDB_C003184 | PGDB_AS000251 | View |
| DC50 | - | = | 1.5 | nM | - | — | GSPT1 | - | NB4 | WO2024222614A1 | PGDB_A035838 | PGDB_C003184 | PGDB_AS001663 | View |
| GI50 | - | = | 13 | nM | - | — | GSPT1 | - | NCI-H1155 | WO2024222614A1 | PGDB_A056085 | PGDB_C003184 | PGDB_AS000187 | View |