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Compound
PGDB_C007963
3 activity records1 related patents
2D structure
O=C1CCC(N2Cc3ccc(CNC(=O)OCc4cnc5c(c4)CCCC5)cc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 10 | uM | - | — | GSPT1 | - | HEK293 | WO2025043225 | PGDB_A017857 | PGDB_C007963 | PGDB_AS002153 | View |
| Dmax | - | = | 52 | % | 10 uM | 6 h | CDK2 | - | HEK293 | WO2025043225 | PGDB_A036534 | PGDB_C007963 | PGDB_AS002435 | View |
| IC50 | - | = | 0.13 | uM | - | — | CDK2 | - | HEK293 | WO2025043225 | PGDB_A062977 | PGDB_C007963 | PGDB_AS002528 | View |