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SIMM · NJU
Assay
PGDB_AS002435
System: cell_based
Target: CDK2
Cell line: HEK293
Assay context summary
Assay context
30 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
Target
CDK2
E3
Not specified
Cell line
HEK293
Technology
luminescence
Activity compounds and values
Activity records
30 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
59
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A017932
PGDB_C007966
PGDB_AS002435
View
Dmax
-
=
12
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A020029
PGDB_C007953
PGDB_AS002435
View
Dmax
-
=
39
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A021055
PGDB_C007935
PGDB_AS002435
View
Dmax
-
=
22
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A024969
PGDB_C007941
PGDB_AS002435
View
Dmax
-
=
21
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A028625
PGDB_C007949
PGDB_AS002435
View
Dmax
-
=
36
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A030969
PGDB_C007936
PGDB_AS002435
View
Dmax
-
=
30
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A034617
PGDB_C007968
PGDB_AS002435
View
Dmax
-
=
52
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A036534
PGDB_C007963
PGDB_AS002435
View
Dmax
-
=
24
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A039489
PGDB_C007943
PGDB_AS002435
View
Dmax
-
=
28
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A040669
PGDB_C007937
PGDB_AS002435
View
Dmax
-
=
35
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A041065
PGDB_C007969
PGDB_AS002435
View
Dmax
-
=
26
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A043841
PGDB_C007965
PGDB_AS002435
View
Dmax
-
=
49
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A046220
PGDB_C007964
PGDB_AS002435
View
Dmax
-
=
30
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A047188
PGDB_C007945
PGDB_AS002435
View
Dmax
-
=
13
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A048011
PGDB_C007944
PGDB_AS002435
View
Dmax
-
=
49
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A051216
PGDB_C007948
PGDB_AS002435
View
Dmax
-
=
52
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A052162
PGDB_C007939
PGDB_AS002435
View
Dmax
-
=
34
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A054566
PGDB_C007942
PGDB_AS002435
View
Dmax
-
=
20
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A056459
PGDB_C007933
PGDB_AS002435
View
Dmax
-
=
21
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A061800
PGDB_C007932
PGDB_AS002435
View