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SIMM · NJU
Assay
PGDB_AS002153
System: cell_based
Target: GSPT1
Cell line: HEK293
Assay context summary
Assay context
16 activity records
Assay family
% Degradation
System
cell_based
Readout
IC50
Target
GSPT1
E3
Not specified
Cell line
HEK293
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
16 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
IC50
-
=
31
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A007981
PGDB_C007932
PGDB_AS002153
View
IC50
-
=
31
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A010214
PGDB_C007947
PGDB_AS002153
View
IC50
-
=
31
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A014467
PGDB_C007938
PGDB_AS002153
View
IC50
-
=
31
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A015897
PGDB_C007951
PGDB_AS002153
View
IC50
-
=
31
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A015982
PGDB_C007936
PGDB_AS002153
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A017857
PGDB_C007963
PGDB_AS002153
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A019731
PGDB_C007969
PGDB_AS002153
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A026105
PGDB_C007964
PGDB_AS002153
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A029882
PGDB_C007966
PGDB_AS002153
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A051785
PGDB_C007967
PGDB_AS002153
View
IC50
-
=
31
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A058252
PGDB_C007948
PGDB_AS002153
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A058369
PGDB_C007968
PGDB_AS002153
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A060084
PGDB_C007965
PGDB_AS002153
View
IC50
-
=
31
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A060880
PGDB_C007937
PGDB_AS002153
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A067710
PGDB_C007962
PGDB_AS002153
View
IC50
-
=
31
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A068962
PGDB_C007939
PGDB_AS002153
View