Assay context summary

Assay context

30 activity records
Activity compounds and values

Activity records

30 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C007944
IC50-=0.36uM-CDK2-HEK293WO2025043225PGDB_A009398PGDB_C007944PGDB_AS002528View
2D structure for PGDB_C007964
IC50-=0.08uM-CDK2-HEK293WO2025043225PGDB_A011000PGDB_C007964PGDB_AS002528View
2D structure for PGDB_C007936
IC50-=0.027uM-CDK2-HEK293WO2025043225PGDB_A012872PGDB_C007936PGDB_AS002528View
2D structure for PGDB_C007942
IC50-=0.16uM-CDK2-HEK293WO2025043225PGDB_A013690PGDB_C007942PGDB_AS002528View
2D structure for PGDB_C007945
IC50-=0.45uM-CDK2-HEK293WO2025043225PGDB_A014045PGDB_C007945PGDB_AS002528View
2D structure for PGDB_C007969
IC50-=0.089uM-CDK2-HEK293WO2025043225PGDB_A017772PGDB_C007969PGDB_AS002528View
2D structure for PGDB_C007934
IC50-=0.48uM-CDK2-HEK293WO2025043225PGDB_A022926PGDB_C007934PGDB_AS002528View
2D structure for PGDB_C007962
IC50-=0.21uM-CDK2-HEK293WO2025043225PGDB_A022975PGDB_C007962PGDB_AS002528View
2D structure for PGDB_C007953
IC50-=0.58uM-CDK2-HEK293WO2025043225PGDB_A023799PGDB_C007953PGDB_AS002528View
2D structure for PGDB_C007952
IC50-=0.46uM-CDK2-HEK293WO2025043225PGDB_A023899PGDB_C007952PGDB_AS002528View
2D structure for PGDB_C007941
IC50-=0.086uM-CDK2-HEK293WO2025043225PGDB_A024593PGDB_C007941PGDB_AS002528View
2D structure for PGDB_C007943
IC50-=0.064uM-CDK2-HEK293WO2025043225PGDB_A026953PGDB_C007943PGDB_AS002528View
2D structure for PGDB_C007950
IC50-=0.32uM-CDK2-HEK293WO2025043225PGDB_A027252PGDB_C007950PGDB_AS002528View
2D structure for PGDB_C007966
IC50-=0.036uM-CDK2-HEK293WO2025043225PGDB_A032341PGDB_C007966PGDB_AS002528View
2D structure for PGDB_C007949
IC50-=0.21uM-CDK2-HEK293WO2025043225PGDB_A034261PGDB_C007949PGDB_AS002528View
2D structure for PGDB_C007937
IC50-=0.36uM-CDK2-HEK293WO2025043225PGDB_A035166PGDB_C007937PGDB_AS002528View
2D structure for PGDB_C007935
IC50-=0.16uM-CDK2-HEK293WO2025043225PGDB_A035971PGDB_C007935PGDB_AS002528View
2D structure for PGDB_C007965
IC50-=0.085uM-CDK2-HEK293WO2025043225PGDB_A037924PGDB_C007965PGDB_AS002528View
2D structure for PGDB_C007947
IC50-=0.22uM-CDK2-HEK293WO2025043225PGDB_A037938PGDB_C007947PGDB_AS002528View
2D structure for PGDB_C007932
IC50-=0.23uM-CDK2-HEK293WO2025043225PGDB_A038133PGDB_C007932PGDB_AS002528View