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SIMM · NJU
Assay
PGDB_AS002528
System: cell_based
Target: CDK2
Cell line: HEK293
Assay context summary
Assay context
30 activity records
Assay family
% Degradation
System
cell_based
Readout
IC50
Target
CDK2
E3
Not specified
Cell line
HEK293
Activity compounds and values
Activity records
30 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
IC50
-
=
0.36
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A009398
PGDB_C007944
PGDB_AS002528
View
IC50
-
=
0.08
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A011000
PGDB_C007964
PGDB_AS002528
View
IC50
-
=
0.027
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A012872
PGDB_C007936
PGDB_AS002528
View
IC50
-
=
0.16
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A013690
PGDB_C007942
PGDB_AS002528
View
IC50
-
=
0.45
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A014045
PGDB_C007945
PGDB_AS002528
View
IC50
-
=
0.089
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A017772
PGDB_C007969
PGDB_AS002528
View
IC50
-
=
0.48
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A022926
PGDB_C007934
PGDB_AS002528
View
IC50
-
=
0.21
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A022975
PGDB_C007962
PGDB_AS002528
View
IC50
-
=
0.58
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A023799
PGDB_C007953
PGDB_AS002528
View
IC50
-
=
0.46
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A023899
PGDB_C007952
PGDB_AS002528
View
IC50
-
=
0.086
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A024593
PGDB_C007941
PGDB_AS002528
View
IC50
-
=
0.064
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A026953
PGDB_C007943
PGDB_AS002528
View
IC50
-
=
0.32
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A027252
PGDB_C007950
PGDB_AS002528
View
IC50
-
=
0.036
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A032341
PGDB_C007966
PGDB_AS002528
View
IC50
-
=
0.21
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A034261
PGDB_C007949
PGDB_AS002528
View
IC50
-
=
0.36
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A035166
PGDB_C007937
PGDB_AS002528
View
IC50
-
=
0.16
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A035971
PGDB_C007935
PGDB_AS002528
View
IC50
-
=
0.085
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A037924
PGDB_C007965
PGDB_AS002528
View
IC50
-
=
0.22
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A037938
PGDB_C007947
PGDB_AS002528
View
IC50
-
=
0.23
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A038133
PGDB_C007932
PGDB_AS002528
View