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Compound
PGDB_C016630
7 activity records1 related patents
2D structure
O=C1CCC(N2C(=O)c3ccc(Br)c4cccc2c34)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Emax | - | > | 60 | % | - | DC50 > 10000 nM | DC50 >= 100 nM and <= 1000 nM | DC50 < 100 nM | - | - | NCI-H929.11 | WO2022081927A1 | PGDB_A013630 | PGDB_C016630 | PGDB_AS001790 | View |
| DC50 | - | > | 10000 | nM | - | — | - | - | NCI-H929.11 | WO2022081927A1 | PGDB_A021854 | PGDB_C016630 | PGDB_AS000877 | View |
| DC50 | - | > | 10000 | nM | - | — | - | - | 293T.114 | WO2022081927A1 | PGDB_A023622 | PGDB_C016630 | PGDB_AS001223 | View |
| Emax | - | < | 45 | % | - | DC50 > 10000 nM | DC50 >= 100 nM and <= 1000 nM | > 100 nM | - | - | KELLY.2 | WO2022081927A1 | PGDB_A040826 | PGDB_C016630 | PGDB_AS000499 | View |
| IC50 | - | = | 40 | nM | - | — | - | - | 293T.116 | WO2022081927A1 | PGDB_A060122 | PGDB_C016630 | PGDB_AS001204 | View |
| Emax | - | > | 60 | % | - | DC50 > 10000 nM | > 100 nM | DC50 < 100 nM | - | - | 293T.114 | WO2022081927A1 | PGDB_A068587 | PGDB_C016630 | PGDB_AS000287 | View |
| DC50 | - | < | 100 | nM | - | — | - | - | KELLY.2 | WO2022081927A1 | PGDB_A073704 | PGDB_C016630 | PGDB_AS001296 | View |