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SIMM · NJU
Assay
PGDB_AS000877
System: cell_based
Target: IKZF1
Cell line: NCI-H929.11
Assay context summary
Assay context
15 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
IKZF1
E3
Not specified
Cell line
NCI-H929.11
Technology
luminescence
Activity compounds and values
Activity records
15 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
>
10000
nM
-
—
-
-
NCI-H929.11
WO2022081927A1
PGDB_A007086
PGDB_C016632
PGDB_AS000877
View
DC50
-
>
10000
nM
-
—
-
-
NCI-H929.11
WO2022081927A1
PGDB_A007258
PGDB_C026783
PGDB_AS000877
View
DC50
-
>
10000
nM
-
—
-
-
NCI-H929.11
WO2022081927A1
PGDB_A010319
PGDB_C026791
PGDB_AS000877
View
DC50
-
>
10000
nM
-
—
-
-
NCI-H929.11
WO2022081927A1
PGDB_A011306
PGDB_C016634
PGDB_AS000877
View
DC50
-
<
100
nM
-
—
-
-
NCI-H929.11
WO2022081927A1
PGDB_A013043
PGDB_C026764
PGDB_AS000877
View
DC50
-
<
100
nM
-
—
-
-
NCI-H929.11
WO2022081927A1
PGDB_A021519
PGDB_C015421
PGDB_AS000877
View
DC50
-
>
10000
nM
-
—
-
-
NCI-H929.11
WO2022081927A1
PGDB_A021854
PGDB_C016630
PGDB_AS000877
View
DC50
-
>
10000
nM
-
—
-
-
NCI-H929.11
WO2022081927A1
PGDB_A037109
PGDB_C016639
PGDB_AS000877
View
DC50
-
>
10000
nM
-
—
-
-
NCI-H929.11
WO2022081927A1
PGDB_A037716
PGDB_C016637
PGDB_AS000877
View
DC50
-
<
100
nM
-
—
-
-
NCI-H929.11
WO2022081927A1
PGDB_A055863
PGDB_C016653
PGDB_AS000877
View
DC50
-
<
100
nM
-
—
-
-
NCI-H929.11
WO2022081927A1
PGDB_A060911
PGDB_C026784
PGDB_AS000877
View
DC50
-
>
10000
nM
-
—
-
-
NCI-H929.11
WO2022081927A1
PGDB_A067984
PGDB_C016644
PGDB_AS000877
View
DC50
-
>
10000
nM
-
—
-
-
NCI-H929.11
WO2022081927A1
PGDB_A070603
PGDB_C016636
PGDB_AS000877
View
DC50
-
>
10000
nM
-
—
-
-
NCI-H929.11
WO2022081927A1
PGDB_A072739
PGDB_C016638
PGDB_AS000877
View
DC50
-
<
100
nM
-
—
-
-
NCI-H929.11
WO2022081927A1
PGDB_A077605
PGDB_C025110
PGDB_AS000877
View