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CCOc1ccc(Cc2ccc3c4c(cccc24)N(C2CCC(=O)NC2=O)C3=O)cc1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Emax | - | > | 60 | % | - | DC50 > 10000 nM | > 100 nM | DC50 < 100 nM | - | - | 293T.114 | WO2022081927A1 | PGDB_A009296 | PGDB_C016638 | PGDB_AS000287 | View | |
| DC50 | - | > | 10000 | nM | - | — | - | - | 293T.114 | WO2022081927A1 | PGDB_A011907 | PGDB_C016638 | PGDB_AS001223 | View | |
| Emax | - | > | 60 | % | - | DC50 > 10000 nM | DC50 >= 100 nM and <= 1000 nM | > 100 nM | - | - | KELLY.2 | WO2022081927A1 | PGDB_A021136 | PGDB_C016638 | PGDB_AS000499 | View | |
| Emax | - | > | 60 | % | - | DC50 > 10000 nM | DC50 >= 100 nM and <= 1000 nM | DC50 < 100 nM | - | - | NCI-H929.11 | WO2022081927A1 | PGDB_A049267 | PGDB_C016638 | PGDB_AS001790 | View | |
| DC50 | - | > | 10000 | nM | - | — | - | - | KELLY.2 | WO2022081927A1 | PGDB_A054985 | PGDB_C016638 | PGDB_AS001296 | View | |
| DC50 | - | > | 10000 | nM | - | — | - | - | NCI-H929.11 | WO2022081927A1 | PGDB_A072739 | PGDB_C016638 | PGDB_AS000877 | View |