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CCOC(=O)c1cc(Cc2ccc3c4c(cccc24)N(C2CCC(=O)NC2=O)C3=O)ccc1F| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | > | 10000 | nM | - | — | - | - | 293T.114 | WO2022081927A1 | PGDB_A014576 | PGDB_C016639 | PGDB_AS001223 | View | |
| Emax | - | > | 60 | % | - | DC50 > 10000 nM | > 100 nM | DC50 < 100 nM | - | - | 293T.114 | WO2022081927A1 | PGDB_A018496 | PGDB_C016639 | PGDB_AS000287 | View | |
| DC50 | - | > | 10000 | nM | - | — | - | - | NCI-H929.11 | WO2022081927A1 | PGDB_A037109 | PGDB_C016639 | PGDB_AS000877 | View | |
| Emax | - | > | 60 | % | - | DC50 > 10000 nM | DC50 >= 100 nM and <= 1000 nM | > 100 nM | - | - | KELLY.2 | WO2022081927A1 | PGDB_A044898 | PGDB_C016639 | PGDB_AS000499 | View | |
| Emax | - | > | 60 | % | - | DC50 > 10000 nM | DC50 >= 100 nM and <= 1000 nM | DC50 < 100 nM | - | - | NCI-H929.11 | WO2022081927A1 | PGDB_A053722 | PGDB_C016639 | PGDB_AS001790 | View | |
| DC50 | - | > | 10000 | nM | - | — | - | - | KELLY.2 | WO2022081927A1 | PGDB_A073970 | PGDB_C016639 | PGDB_AS001296 | View |