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Compound
PGDB_C020479
7 activity records1 related patents
2D structure
CCC(=O)Nc1ccc(COC(=O)N(C)CC(C)(C)COCCc2ccc(C(=O)NCc3ccc4c5c(cccc35)C(=O)N4C3CCC(=O)NC3=O)cc2Cl)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Selectivity index | 293T/HCC569 | = | 10-100 | fold | - | — | - | - | - | WO2025162410A1 | PGDB_A016034 | PGDB_C020479 | PGDB_AS000299 | View |
| IC50 | - | = | <= 0.5 | nM | - | — | GSPT1 | - | HEK293T | WO2025162410A1 | PGDB_A026467 | PGDB_C020479 | PGDB_AS002143 | View |
| Selectivity index | 293T/HCC569 | = | 10-100 | fold | - | — | - | - | - | WO2025162410A1 | PGDB_A029445 | PGDB_C020479 | PGDB_AS000299 | View |
| IC50 | - | <= | 0.5 | nM | - | — | GSPT1 | - | HCC1569 | WO2025162410A1 | PGDB_A044846 | PGDB_C020479 | PGDB_AS001676 | View |
| EC50 | - | = | <= 0.5 | nM | - | — | GSPT1 | - | - | WO2025162410A1 | PGDB_A056919 | PGDB_C020479 | PGDB_AS002258 | View |
| EC50 | - | = | <= 0.5 | nM | - | — | GSPT1 | - | - | WO2025162410A1 | PGDB_A058579 | PGDB_C020479 | PGDB_AS002258 | View |
| IC50 | - | = | <= 0.5 | nM | - | — | GSPT1 | - | HEK293T | WO2025162410A1 | PGDB_A065606 | PGDB_C020479 | PGDB_AS002143 | View |