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SIMM · NJU
Assay
PGDB_AS000307
System: biochemical
Target: RAF1
Assay context summary
Assay context
45 activity records
Assay family
biochemical
System
biochemical
Readout
IC50
Target
RAF1
E3
Not specified
Technology
HTRF
Activity compounds and values
Activity records
45 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A008927
PGDB_C011589
PGDB_AS000307
View
IC50
-
=
100-1000
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A010312
PGDB_C011622
PGDB_AS000307
View
IC50
-
=
100-1000
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A010959
PGDB_C011593
PGDB_AS000307
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A012757
PGDB_C011618
PGDB_AS000307
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A014079
PGDB_C011620
PGDB_AS000307
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A014446
PGDB_C011625
PGDB_AS000307
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A016221
PGDB_C011599
PGDB_AS000307
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A016578
PGDB_C011602
PGDB_AS000307
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A019709
PGDB_C011591
PGDB_AS000307
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A020417
PGDB_C011624
PGDB_AS000307
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A020711
PGDB_C011628
PGDB_AS000307
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A020900
PGDB_C011605
PGDB_AS000307
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A021835
PGDB_C011601
PGDB_AS000307
View
IC50
-
=
100-1000
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A022801
PGDB_C011588
PGDB_AS000307
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A022888
PGDB_C011629
PGDB_AS000307
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A024296
PGDB_C011592
PGDB_AS000307
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A024418
PGDB_C011587
PGDB_AS000307
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A025935
PGDB_C011627
PGDB_AS000307
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A026533
PGDB_C011608
PGDB_AS000307
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A030859
PGDB_C011598
PGDB_AS000307
View