Assay

PGDB_AS000322

System: cell_basedTarget: GSPT1Cell line: HEK293T
Assay context summary

Assay context

21 activity records
Assay family% Degradation
Systemcell_based
ReadoutDC50
TargetGSPT1
E3Not specified
Cell lineHEK293T
Technologyluminescence
Activity compounds and values

Activity records

21 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C000471
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A007005PGDB_C000471PGDB_AS000322View
2D structure for PGDB_C000472
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A007616PGDB_C000472PGDB_AS000322View
2D structure for PGDB_C000470
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A012140PGDB_C000470PGDB_AS000322View
2D structure for PGDB_C000392
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A018789PGDB_C000392PGDB_AS000322View
2D structure for PGDB_C000464
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A022364PGDB_C000464PGDB_AS000322View
2D structure for PGDB_C000466
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A024731PGDB_C000466PGDB_AS000322View
2D structure for PGDB_C000469
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A030309PGDB_C000469PGDB_AS000322View
2D structure for PGDB_C000401
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A033337PGDB_C000401PGDB_AS000322View
2D structure for PGDB_C000414
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A036836PGDB_C000414PGDB_AS000322View
2D structure for PGDB_C000413
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A043683PGDB_C000413PGDB_AS000322View
2D structure for PGDB_C000463
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A046653PGDB_C000463PGDB_AS000322View
2D structure for PGDB_C000414
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A050116PGDB_C000414PGDB_AS000322View
2D structure for PGDB_C000391
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A056146PGDB_C000391PGDB_AS000322View
2D structure for PGDB_C000381
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A056824PGDB_C000381PGDB_AS000322View
2D structure for PGDB_C000453
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A057394PGDB_C000453PGDB_AS000322View
2D structure for PGDB_C000466
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A059261PGDB_C000466PGDB_AS000322View
2D structure for PGDB_C000390
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A061214PGDB_C000390PGDB_AS000322View
2D structure for PGDB_C000468
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A065559PGDB_C000468PGDB_AS000322View
2D structure for PGDB_C000402
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A069342PGDB_C000402PGDB_AS000322View
2D structure for PGDB_C000387
DC50->30uM-—GSPT1-HEK293TUS20230265071A1PGDB_A073535PGDB_C000387PGDB_AS000322View
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