Assay
PGDB_AS000327
System: cell_basedCell line: NCI-H929
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 60 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | - | - | NCI-H929 | EP4685141A1 | PGDB_A017131 | PGDB_C025619 | PGDB_AS000327 | View | |
| Dmax | - | = | 65.3 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | - | - | NCI-H929 | EP4685141A1 | PGDB_A022618 | PGDB_C025616 | PGDB_AS000327 | View | |
| Dmax | - | = | 75.8 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | - | - | NCI-H929 | EP4685141A1 | PGDB_A052443 | PGDB_C025597 | PGDB_AS000327 | View | |
| Dmax | - | = | 68.4 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | - | - | NCI-H929 | EP4685141A1 | PGDB_A058075 | PGDB_C025601 | PGDB_AS000327 | View | |
| Dmax | - | = | 65.8 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | - | - | NCI-H929 | EP4685141A1 | PGDB_A060861 | PGDB_C025617 | PGDB_AS000327 | View | |
| Dmax | - | = | 74.1 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | - | - | NCI-H929 | EP4685141A1 | PGDB_A061356 | PGDB_C025624 | PGDB_AS000327 | View | |
| Dmax | - | = | 77 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | - | - | NCI-H929 | EP4685141A1 | PGDB_A063874 | PGDB_C025625 | PGDB_AS000327 | View | |
| Dmax | - | = | 73.6 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | - | - | NCI-H929 | EP4685141A1 | PGDB_A070490 | PGDB_C025600 | PGDB_AS000327 | View | |
| Dmax | - | = | 73.6 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | - | - | NCI-H929 | EP4685141A1 | PGDB_A073830 | PGDB_C025599 | PGDB_AS000327 | View | |
| Dmax | - | = | 57.1 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | - | - | NCI-H929 | EP4685141A1 | PGDB_A074876 | PGDB_C025615 | PGDB_AS000327 | View |