PatGlueDB | Molecular Glue Patent Bioactivity Database

Patent summary

Publication numberEP4685141A1

AssigneeShanghai Helioson Pharmaceutical

Family members4

Filing year2,024

JurisdictionEP

Compounds78

Activity records143

Assays9

Activity compounds and values

Activity records

143 records

	Control		Value		Concentration	Time				Record ID	Compound	Assay	Details
IC50	-	=	0.03	nM	-	—	-	-	NCI-H929	PGDB_A007771	PGDB_C025659	PGDB_AS001501	View
IC50	-	=	0.01	nM	-	—	-	-	NCI-H929	PGDB_A008329	PGDB_C025614	PGDB_AS001501	View
DC50	-	=	0.081	nM	-	—	-	-	NCI-H929	PGDB_A008886	PGDB_C025599	PGDB_AS001024	View
DC50	-	=	0.37	nM	-	—	-	-	NCI-H929	PGDB_A009501	PGDB_C025624	PGDB_AS001024	View
IC50	-	=	0.01	nM	-	—	-	-	NCI-H929	PGDB_A010130	PGDB_C025638	PGDB_AS001501	View
IC50	-	=	27	nM	-	—	-	-	-	PGDB_A011053	PGDB_C025624	PGDB_AS001840	View
IC50	-	=	0.01	nM	-	—	-	-	NCI-H929	PGDB_A011493	PGDB_C025636	PGDB_AS001501	View
IC50	-	=	1.6	nM	-	—	-	-	NCI-H929	PGDB_A012192	PGDB_C025672	PGDB_AS001501	View
IC50	-	=	0.07	nM	-	—	-	-	NCI-H929	PGDB_A012215	PGDB_C025656	PGDB_AS001501	View
IC50	-	=	0.07	nM	-	—	-	-	NCI-H929	PGDB_A012997	PGDB_C025609	PGDB_AS001501	View
Dmax	-	=	70.3	%	Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM	24 h	-	-	NCI-H929	PGDB_A013216	PGDB_C025600	PGDB_AS002256	View
IC50	-	=	0.02	nM	-	—	-	-	NCI-H929	PGDB_A013723	PGDB_C025674	PGDB_AS001501	View
IC50	-	=	20	nM	-	—	-	-	-	PGDB_A013775	PGDB_C025616	PGDB_AS001840	View
Dmax	-	=	76.6	%	Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM	24 h	-	-	NCI-H929	PGDB_A014505	PGDB_C025599	PGDB_AS002256	View
IC50	-	=	0.01	nM	-	—	-	-	NCI-H929	PGDB_A014585	PGDB_C025645	PGDB_AS001501	View
Dmax	-	=	74.1	%	Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM	24 h	-	-	NCI-H929	PGDB_A014693	PGDB_C025615	PGDB_AS002256	View
IC50	-	=	0.01	nM	-	—	-	-	NCI-H929	PGDB_A015092	PGDB_C025634	PGDB_AS001501	View
IC50	-	=	0.01	nM	-	—	-	-	NCI-H929	PGDB_A015343	PGDB_C025617	PGDB_AS001501	View
IC50	-	=	34	nM	-	—	-	-	-	PGDB_A016448	PGDB_C025615	PGDB_AS001275	View
Dmax	-	=	60	%	Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM	24 h	-	-	NCI-H929	PGDB_A017131	PGDB_C025619	PGDB_AS000327	View

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