Assay
PGDB_AS000575
System: cell_basedCell line: NCI-H929
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 0.05 | nM | - | — | - | - | NCI-H929 | EP4685141A1 | PGDB_A023239 | PGDB_C025599 | PGDB_AS000575 | View | |
| DC50 | - | = | 0.093 | nM | - | — | - | - | NCI-H929 | EP4685141A1 | PGDB_A023820 | PGDB_C025624 | PGDB_AS000575 | View | |
| DC50 | - | = | 0.22 | nM | - | — | - | - | NCI-H929 | EP4685141A1 | PGDB_A026595 | PGDB_C025615 | PGDB_AS000575 | View | |
| DC50 | - | = | 0.075 | nM | - | — | - | - | NCI-H929 | EP4685141A1 | PGDB_A039811 | PGDB_C025619 | PGDB_AS000575 | View | |
| DC50 | - | = | 0.12 | nM | - | — | - | - | NCI-H929 | EP4685141A1 | PGDB_A044865 | PGDB_C025597 | PGDB_AS000575 | View | |
| DC50 | - | = | 0.12 | nM | - | — | - | - | NCI-H929 | EP4685141A1 | PGDB_A046148 | PGDB_C025601 | PGDB_AS000575 | View | |
| DC50 | - | = | 0.036 | nM | - | — | - | - | NCI-H929 | EP4685141A1 | PGDB_A056641 | PGDB_C025617 | PGDB_AS000575 | View | |
| DC50 | - | = | 0.056 | nM | - | — | - | - | NCI-H929 | EP4685141A1 | PGDB_A070471 | PGDB_C025616 | PGDB_AS000575 | View | |
| DC50 | - | = | 0.16 | nM | - | — | - | - | NCI-H929 | EP4685141A1 | PGDB_A074411 | PGDB_C025625 | PGDB_AS000575 | View | |
| DC50 | - | = | 0.19 | nM | - | — | - | - | NCI-H929 | EP4685141A1 | PGDB_A074950 | PGDB_C025600 | PGDB_AS000575 | View |