Assay context summary

Assay context

58 activity records
Activity compounds and values

Activity records

58 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C019219
IC50-<1nM-IKZF3-JurkatWO2025016359A1PGDB_A007321PGDB_C019219PGDB_AS000690View
2D structure for PGDB_C019203
IC50-=10-50nM-IKZF3-JurkatWO2025016359A1PGDB_A010499PGDB_C019203PGDB_AS000690View
2D structure for PGDB_C019199
IC50-=1-5nM-IKZF3-JurkatWO2025016359A1PGDB_A011077PGDB_C019199PGDB_AS000690View
2D structure for PGDB_C019256
IC50-<1nM-IKZF3-JurkatWO2025016359A1PGDB_A013200PGDB_C019256PGDB_AS000690View
2D structure for PGDB_C019196
IC50-=5-10nM-IKZF3-JurkatWO2025016359A1PGDB_A014506PGDB_C019196PGDB_AS000690View
2D structure for PGDB_C019228
IC50-=10-50nM-IKZF3-JurkatWO2025016359A1PGDB_A015641PGDB_C019228PGDB_AS000690View
2D structure for PGDB_C019247
IC50-=50-100nM-IKZF3-JurkatWO2025016359A1PGDB_A015853PGDB_C019247PGDB_AS000690View
2D structure for PGDB_C019204
IC50-=1-5nM-IKZF3-JurkatWO2025016359A1PGDB_A016197PGDB_C019204PGDB_AS000690View
2D structure for PGDB_C019187
IC50-=100-500nM-IKZF3-JurkatWO2025016359A1PGDB_A018522PGDB_C019187PGDB_AS000690View
2D structure for PGDB_C019188
IC50-=1-5nM-IKZF3-JurkatWO2025016359A1PGDB_A018752PGDB_C019188PGDB_AS000690View
2D structure for PGDB_C019175
IC50-=1-5nM-IKZF3-JurkatWO2025016359A1PGDB_A019017PGDB_C019175PGDB_AS000690View
2D structure for PGDB_C019195
IC50-=1-5nM-IKZF3-JurkatWO2025016359A1PGDB_A019301PGDB_C019195PGDB_AS000690View
2D structure for PGDB_C019181
IC50-=1-5nM-IKZF3-JurkatWO2025016359A1PGDB_A020354PGDB_C019181PGDB_AS000690View
2D structure for PGDB_C019201
IC50-=5-10nM-IKZF3-JurkatWO2025016359A1PGDB_A022442PGDB_C019201PGDB_AS000690View
2D structure for PGDB_C019260
IC50-=10-50nM-IKZF3-JurkatWO2025016359A1PGDB_A023391PGDB_C019260PGDB_AS000690View
2D structure for PGDB_C019216
IC50-=5-10nM-IKZF3-JurkatWO2025016359A1PGDB_A025887PGDB_C019216PGDB_AS000690View
2D structure for PGDB_C019193
IC50-=5-10nM-IKZF3-JurkatWO2025016359A1PGDB_A026628PGDB_C019193PGDB_AS000690View
2D structure for PGDB_C019220
IC50-=5-10nM-IKZF3-JurkatWO2025016359A1PGDB_A026899PGDB_C019220PGDB_AS000690View
2D structure for PGDB_C019176
IC50-=1-5nM-IKZF3-JurkatWO2025016359A1PGDB_A026961PGDB_C019176PGDB_AS000690View
2D structure for PGDB_C019255
IC50-=5-10nM-IKZF3-JurkatWO2025016359A1PGDB_A029620PGDB_C019255PGDB_AS000690View