Assay
PGDB_AS000833
System: cell_basedTarget: IKZF1Cell line: NCI-H929
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
 | Dmax | - | = | 73.6 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF1 | - | NCI-H929 | CA3286762A1 | PGDB_A007207 | PGDB_C025599 | PGDB_AS000833 | View |
 | Dmax | - | = | 65.3 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF1 | - | NCI-H929 | CA3286762A1 | PGDB_A015525 | PGDB_C025616 | PGDB_AS000833 | View |
 | Dmax | - | = | 57.1 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF1 | - | NCI-H929 | CA3286762A1 | PGDB_A017018 | PGDB_C025615 | PGDB_AS000833 | View |
 | Dmax | - | = | 74.1 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF1 | - | NCI-H929 | CA3286762A1 | PGDB_A017888 | PGDB_C021277 | PGDB_AS000833 | View |
 | Dmax | - | = | 68.4 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF1 | - | NCI-H929 | CA3286762A1 | PGDB_A031892 | PGDB_C025601 | PGDB_AS000833 | View |
 | Dmax | - | = | 77 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF1 | - | NCI-H929 | CA3286762A1 | PGDB_A034585 | PGDB_C021276 | PGDB_AS000833 | View |
 | Dmax | - | = | 60 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF1 | - | NCI-H929 | CA3286762A1 | PGDB_A043944 | PGDB_C025619 | PGDB_AS000833 | View |
 | Dmax | - | = | 75.8 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF1 | - | NCI-H929 | CA3286762A1 | PGDB_A045394 | PGDB_C025597 | PGDB_AS000833 | View |
 | Dmax | - | = | 65.8 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF1 | - | NCI-H929 | CA3286762A1 | PGDB_A047362 | PGDB_C025617 | PGDB_AS000833 | View |
 | Dmax | - | = | 73.6 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF1 | - | NCI-H929 | CA3286762A1 | PGDB_A052714 | PGDB_C025600 | PGDB_AS000833 | View |