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SIMM · NJU
Assay
PGDB_AS001026
System: cell_based
Cell line: MV-4-11
Assay context summary
Assay context
16 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
E3
Not specified
Cell line
MV-4-11
Technology
Western_blot
Detection target
protein_degradation
Activity compounds and values
Activity records
16 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
<
10
nM
-
—
CSNK1A1
-
MV-4-11
CN121471230A
PGDB_A009050
PGDB_C001054
PGDB_AS001026
View
DC50
-
<
10
nM
-
—
CSNK1A1
-
MV-4-11
CN121471230A
PGDB_A011335
PGDB_C001061
PGDB_AS001026
View
DC50
-
<
10
nM
-
—
CSNK1A1
-
MV-4-11
CN121471230A
PGDB_A011590
PGDB_C001059
PGDB_AS001026
View
DC50
-
<
10
nM
-
—
CSNK1A1
-
MV-4-11
CN121471230A
PGDB_A017726
PGDB_C001060
PGDB_AS001026
View
DC50
-
<
10
nM
-
—
CSNK1A1
-
MV-4-11
CN121471230A
PGDB_A038188
PGDB_C001050
PGDB_AS001026
View
DC50
-
<
10
nM
-
—
CSNK1A1
-
MV-4-11
CN121471230A
PGDB_A039309
PGDB_C001052
PGDB_AS001026
View
DC50
-
<
10
nM
-
—
CSNK1A1
-
MV-4-11
CN121471230A
PGDB_A042870
PGDB_C001058
PGDB_AS001026
View
DC50
-
<
10
nM
-
—
CSNK1A1
-
MV-4-11
CN121471230A
PGDB_A044349
PGDB_C001062
PGDB_AS001026
View
DC50
-
<
10
nM
-
—
CSNK1A1
-
MV-4-11
CN121471230A
PGDB_A046394
PGDB_C001051
PGDB_AS001026
View
DC50
-
<
10
nM
-
—
CSNK1A1
-
MV-4-11
CN121471230A
PGDB_A053113
PGDB_C001056
PGDB_AS001026
View
DC50
-
<
10
nM
-
—
CSNK1A1
-
MV-4-11
CN121471230A
PGDB_A059496
PGDB_C001048
PGDB_AS001026
View
DC50
-
<
10
nM
-
—
CSNK1A1
-
MV-4-11
CN121471230A
PGDB_A060355
PGDB_C001053
PGDB_AS001026
View
DC50
-
<
10
nM
-
—
CSNK1A1
-
MV-4-11
CN121471230A
PGDB_A062361
PGDB_C001049
PGDB_AS001026
View
DC50
-
<
10
nM
-
—
CSNK1A1
-
MV-4-11
CN121471230A
PGDB_A062827
PGDB_C001046
PGDB_AS001026
View
DC50
-
<
10
nM
-
—
CSNK1A1
-
MV-4-11
CN121471230A
PGDB_A073775
PGDB_C001063
PGDB_AS001026
View
DC50
-
<
10
nM
-
—
CSNK1A1
-
MV-4-11
CN121471230A
PGDB_A077879
PGDB_C001057
PGDB_AS001026
View