Assay
PGDB_AS001203
System: cell_basedCell line: AsPC-1
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 1.764 | nM | - | — | KRAS | - | AsPC-1 | CN121181579A | PGDB_A017494 | PGDB_C024605 | PGDB_AS001203 | View | |
| IC50 | - | = | 2.496 | nM | - | — | KRAS | - | AsPC-1 | CN121181579A | PGDB_A032413 | PGDB_C011631 | PGDB_AS001203 | View | |
| IC50 | - | = | 0.3578 | nM | - | — | KRAS | - | AsPC-1 | CN121181579A | PGDB_A043590 | PGDB_C024673 | PGDB_AS001203 | View | |
| IC50 | - | = | 7.456 | nM | - | — | KRAS | - | AsPC-1 | CN121181579A | PGDB_A051912 | PGDB_C011587 | PGDB_AS001203 | View | |
| IC50 | - | = | 0.9378 | nM | - | — | KRAS | - | AsPC-1 | CN121181579A | PGDB_A068037 | PGDB_C024617 | PGDB_AS001203 | View | |
| IC50 | - | = | 1.579 | nM | - | — | KRAS | - | AsPC-1 | CN121181579A | PGDB_A069727 | PGDB_C024627 | PGDB_AS001203 | View |