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SIMM · NJU
Assay
PGDB_AS001302
System: cell_based
Target: CDK2
Cell line: HEK293
Assay context summary
Assay context
50 activity records
Assay family
% Degradation
System
cell_based
Readout
IC50
Target
CDK2
E3
Not specified
Cell line
HEK293
Activity compounds and values
Activity records
50 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
IC50
-
=
0.0078
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A013325
PGDB_C007999
PGDB_AS001302
View
IC50
-
=
0.012
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A014451
PGDB_C008001
PGDB_AS001302
View
IC50
-
=
0.0062
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A017762
PGDB_C007981
PGDB_AS001302
View
IC50
-
=
0.047
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A020420
PGDB_C007974
PGDB_AS001302
View
IC50
-
=
0.051
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A022034
PGDB_C007994
PGDB_AS001302
View
IC50
-
=
0.051
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A022538
PGDB_C007983
PGDB_AS001302
View
IC50
-
=
0.14
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A024452
PGDB_C007993
PGDB_AS001302
View
IC50
-
=
0.34
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A026309
PGDB_C007985
PGDB_AS001302
View
IC50
-
=
0.011
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A029883
PGDB_C008009
PGDB_AS001302
View
IC50
-
=
0.046
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A031865
PGDB_C007996
PGDB_AS001302
View
IC50
-
=
0.035
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A032489
PGDB_C007988
PGDB_AS001302
View
IC50
-
=
0.14
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A032594
PGDB_C007992
PGDB_AS001302
View
IC50
-
=
0.087
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A034047
PGDB_C007977
PGDB_AS001302
View
IC50
-
=
0.11
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A034446
PGDB_C007975
PGDB_AS001302
View
IC50
-
=
0.14
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A038476
PGDB_C008018
PGDB_AS001302
View
IC50
-
=
0.13
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A038815
PGDB_C007971
PGDB_AS001302
View
IC50
-
=
0.048
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A040396
PGDB_C008006
PGDB_AS001302
View
IC50
-
=
0.023
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A041531
PGDB_C008007
PGDB_AS001302
View
IC50
-
=
0.028
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A045008
PGDB_C007972
PGDB_AS001302
View
IC50
-
=
0.036
uM
-
—
CDK2
-
HEK293
WO2025043225
PGDB_A045202
PGDB_C007991
PGDB_AS001302
View