Assay context summary

Assay context

50 activity records
Activity compounds and values

Activity records

50 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C007999
IC50-=0.0078uM-CDK2-HEK293WO2025043225PGDB_A013325PGDB_C007999PGDB_AS001302View
2D structure for PGDB_C008001
IC50-=0.012uM-CDK2-HEK293WO2025043225PGDB_A014451PGDB_C008001PGDB_AS001302View
2D structure for PGDB_C007981
IC50-=0.0062uM-CDK2-HEK293WO2025043225PGDB_A017762PGDB_C007981PGDB_AS001302View
2D structure for PGDB_C007974
IC50-=0.047uM-CDK2-HEK293WO2025043225PGDB_A020420PGDB_C007974PGDB_AS001302View
2D structure for PGDB_C007994
IC50-=0.051uM-CDK2-HEK293WO2025043225PGDB_A022034PGDB_C007994PGDB_AS001302View
2D structure for PGDB_C007983
IC50-=0.051uM-CDK2-HEK293WO2025043225PGDB_A022538PGDB_C007983PGDB_AS001302View
2D structure for PGDB_C007993
IC50-=0.14uM-CDK2-HEK293WO2025043225PGDB_A024452PGDB_C007993PGDB_AS001302View
2D structure for PGDB_C007985
IC50-=0.34uM-CDK2-HEK293WO2025043225PGDB_A026309PGDB_C007985PGDB_AS001302View
2D structure for PGDB_C008009
IC50-=0.011uM-CDK2-HEK293WO2025043225PGDB_A029883PGDB_C008009PGDB_AS001302View
2D structure for PGDB_C007996
IC50-=0.046uM-CDK2-HEK293WO2025043225PGDB_A031865PGDB_C007996PGDB_AS001302View
2D structure for PGDB_C007988
IC50-=0.035uM-CDK2-HEK293WO2025043225PGDB_A032489PGDB_C007988PGDB_AS001302View
2D structure for PGDB_C007992
IC50-=0.14uM-CDK2-HEK293WO2025043225PGDB_A032594PGDB_C007992PGDB_AS001302View
2D structure for PGDB_C007977
IC50-=0.087uM-CDK2-HEK293WO2025043225PGDB_A034047PGDB_C007977PGDB_AS001302View
2D structure for PGDB_C007975
IC50-=0.11uM-CDK2-HEK293WO2025043225PGDB_A034446PGDB_C007975PGDB_AS001302View
2D structure for PGDB_C008018
IC50-=0.14uM-CDK2-HEK293WO2025043225PGDB_A038476PGDB_C008018PGDB_AS001302View
2D structure for PGDB_C007971
IC50-=0.13uM-CDK2-HEK293WO2025043225PGDB_A038815PGDB_C007971PGDB_AS001302View
2D structure for PGDB_C008006
IC50-=0.048uM-CDK2-HEK293WO2025043225PGDB_A040396PGDB_C008006PGDB_AS001302View
2D structure for PGDB_C008007
IC50-=0.023uM-CDK2-HEK293WO2025043225PGDB_A041531PGDB_C008007PGDB_AS001302View
2D structure for PGDB_C007972
IC50-=0.028uM-CDK2-HEK293WO2025043225PGDB_A045008PGDB_C007972PGDB_AS001302View
2D structure for PGDB_C007991
IC50-=0.036uM-CDK2-HEK293WO2025043225PGDB_A045202PGDB_C007991PGDB_AS001302View