Assay

PGDB_AS001357

System: cell_basedTarget: BRD4Cell line: HL-60
Assay context summary

Assay context

22 activity records
Assay familyviability
Systemcell_based
ReadoutIC50
TargetBRD4
E3Not specified
Cell lineHL-60
Activity compounds and values

Activity records

22 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C000361
IC50-=100-1000nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A007022PGDB_C000361PGDB_AS001357View
2D structure for PGDB_C000368
IC50-<100nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A008239PGDB_C000368PGDB_AS001357View
2D structure for PGDB_C000376
IC50-<100nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A014248PGDB_C000376PGDB_AS001357View
2D structure for PGDB_C000363
IC50-=100-1000nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A023188PGDB_C000363PGDB_AS001357View
2D structure for PGDB_C000364
IC50-=55nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A025822PGDB_C000364PGDB_AS001357View
2D structure for PGDB_C000366
IC50-<100nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A028497PGDB_C000366PGDB_AS001357View
2D structure for PGDB_C000370
IC50-<100nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A028905PGDB_C000370PGDB_AS001357View
2D structure for PGDB_C000374
IC50-=7.4nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A031117PGDB_C000374PGDB_AS001357View
2D structure for PGDB_C000369
IC50-<100nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A035580PGDB_C000369PGDB_AS001357View
2D structure for PGDB_C000367
IC50-<100nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A037215PGDB_C000367PGDB_AS001357View
2D structure for PGDB_C000359
IC50-=100-1000nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A047483PGDB_C000359PGDB_AS001357View
2D structure for PGDB_C000373
IC50-=8.8nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A050513PGDB_C000373PGDB_AS001357View
2D structure for PGDB_C000377
IC50-=100-1000nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A050817PGDB_C000377PGDB_AS001357View
2D structure for PGDB_C000372
IC50-=12.4nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A054737PGDB_C000372PGDB_AS001357View
2D structure for PGDB_C000365
IC50-<100nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A056321PGDB_C000365PGDB_AS001357View
2D structure for PGDB_C000360
IC50-=100-1000nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A058544PGDB_C000360PGDB_AS001357View
2D structure for PGDB_C000375
IC50-<100nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A059704PGDB_C000375PGDB_AS001357View
2D structure for PGDB_C000371
IC50-<100nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A061933PGDB_C000371PGDB_AS001357View
2D structure for PGDB_C000379
IC50-=1000-2000nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A062394PGDB_C000379PGDB_AS001357View
2D structure for PGDB_C000362
IC50-=100-1000nM-—BRD4/GSPT1-HL-60CN117756818APGDB_A067491PGDB_C000362PGDB_AS001357View
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