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SIMM · NJU
Assay
PGDB_AS001378
System: cell_based
Target: GSPT1
Cell line: HEK293T
Assay context summary
Assay context
21 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
GSPT1
E3
Not specified
Cell line
HEK293T
Detection target
protein_degradation
Activity compounds and values
Activity records
21 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A007308
PGDB_C000401
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A011997
PGDB_C000414
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A014258
PGDB_C000466
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A017118
PGDB_C000392
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A020044
PGDB_C000380
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A020429
PGDB_C000464
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A023504
PGDB_C000391
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A024274
PGDB_C000413
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A030034
PGDB_C000466
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A038641
PGDB_C000472
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A046375
PGDB_C000414
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A048650
PGDB_C000471
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A050022
PGDB_C000381
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A052254
PGDB_C000402
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A052391
PGDB_C000470
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A053463
PGDB_C000463
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A055658
PGDB_C000453
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A058559
PGDB_C000390
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A059021
PGDB_C000469
PGDB_AS001378
View
DC50
-
>
30
uM
-
—
GSPT1
-
HEK293T
CN117836288A
PGDB_A069531
PGDB_C000468
PGDB_AS001378
View