Assay

PGDB_AS001462

System: cell_basedTarget: CRBN
Assay context summary

Assay context

143 activity records
Assay familybiochemical
Systemcell_based
Readout% Inhibition
TargetCRBN
E3CRBN
TechnologyHTRF
Detection targetcell_inhibition
Activity compounds and values

Activity records

143 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C000743
% Inhibition-=53-60%2 uM-CRBNCRBN-CN120548310APGDB_A009157PGDB_C000743PGDB_AS001462View
2D structure for PGDB_C000897
% Inhibition-=40-53%2 uM-CRBNCRBN-CN120548310APGDB_A009265PGDB_C000897PGDB_AS001462View
2D structure for PGDB_C000978
% Inhibition-=70-80%2 uM-CRBNCRBN-CN120548310APGDB_A009414PGDB_C000978PGDB_AS001462View
2D structure for PGDB_C000829
% Inhibition-=70-80%2 uM-CRBNCRBN-CN120548310APGDB_A012016PGDB_C000829PGDB_AS001462View
2D structure for PGDB_C000947
% Inhibition-=53-60%2 uM-CRBNCRBN-CN120548310APGDB_A012598PGDB_C000947PGDB_AS001462View
2D structure for PGDB_C000863
% Inhibition-=53-60%2 uM-CRBNCRBN-CN120548310APGDB_A014376PGDB_C000863PGDB_AS001462View
2D structure for PGDB_C000875
% Inhibition-=40-53%2 uM-CRBNCRBN-CN120548310APGDB_A014854PGDB_C000875PGDB_AS001462View
2D structure for PGDB_C000884
% Inhibition-=53-60%2 uM-CRBNCRBN-CN120548310APGDB_A015126PGDB_C000884PGDB_AS001462View
2D structure for PGDB_C000847
% Inhibition-=53-60%2 uM-CRBNCRBN-CN120548310APGDB_A015336PGDB_C000847PGDB_AS001462View
2D structure for PGDB_C000977
% Inhibition-=70-80%2 uM-CRBNCRBN-CN120548310APGDB_A015886PGDB_C000977PGDB_AS001462View
2D structure for PGDB_C000798
% Inhibition-=70-80%2 uM-CRBNCRBN-CN120548310APGDB_A016242PGDB_C000798PGDB_AS001462View
2D structure for PGDB_C000844
% Inhibition-=40-53%2 uM-CRBNCRBN-CN120548310APGDB_A018259PGDB_C000844PGDB_AS001462View
2D structure for PGDB_C000802
% Inhibition-=70-80%2 uM-CRBNCRBN-CN120548310APGDB_A018327PGDB_C000802PGDB_AS001462View
2D structure for PGDB_C000905
% Inhibition-=40-53%2 uM-CRBNCRBN-CN120548310APGDB_A019396PGDB_C000905PGDB_AS001462View
2D structure for PGDB_C000855
% Inhibition-=70-80%2 uM-CRBNCRBN-CN120548310APGDB_A019512PGDB_C000855PGDB_AS001462View
2D structure for PGDB_C000820
% Inhibition-=70-80%2 uM-CRBNCRBN-CN120548310APGDB_A019983PGDB_C000820PGDB_AS001462View
2D structure for PGDB_C000832
% Inhibition-=40-53%2 uM-CRBNCRBN-CN120548310APGDB_A020291PGDB_C000832PGDB_AS001462View
2D structure for PGDB_C000856
% Inhibition-=70-80%2 uM-CRBNCRBN-CN120548310APGDB_A020749PGDB_C000856PGDB_AS001462View
2D structure for PGDB_C000934
% Inhibition-=60-70%2 uM-CRBNCRBN-CN120548310APGDB_A021048PGDB_C000934PGDB_AS001462View
2D structure for PGDB_C000941
% Inhibition-=70-80%2 uM-CRBNCRBN-CN120548310APGDB_A021489PGDB_C000941PGDB_AS001462View
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