Assay context summary

Assay context

26 activity records
Activity compounds and values

Activity records

26 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C019212
IC50-=50-100nM-IKZF3-MGC-803WO2025016359A1PGDB_A011107PGDB_C019212PGDB_AS001973View
2D structure for PGDB_C019176
IC50-=10-50nM-IKZF3-MGC-803WO2025016359A1PGDB_A015575PGDB_C019176PGDB_AS001973View
2D structure for PGDB_C019195
IC50-=50-100nM-IKZF3-MGC-803WO2025016359A1PGDB_A015975PGDB_C019195PGDB_AS001973View
2D structure for PGDB_C019175
IC50-=10-50nM-IKZF3-MGC-803WO2025016359A1PGDB_A017258PGDB_C019175PGDB_AS001973View
2D structure for PGDB_C019182
IC50-=50-100nM-IKZF3-MGC-803WO2025016359A1PGDB_A017602PGDB_C019182PGDB_AS001973View
2D structure for PGDB_C019201
IC50-=500-1000nM-IKZF3-MGC-803WO2025016359A1PGDB_A017790PGDB_C019201PGDB_AS001973View
2D structure for PGDB_C019199
IC50-=50-100nM-IKZF3-MGC-803WO2025016359A1PGDB_A022917PGDB_C019199PGDB_AS001973View
2D structure for PGDB_C019218
IC50-=10-50nM-IKZF3-MGC-803WO2025016359A1PGDB_A023748PGDB_C019218PGDB_AS001973View
2D structure for PGDB_C019177
IC50-=100-500nM-IKZF3-MGC-803WO2025016359A1PGDB_A023968PGDB_C019177PGDB_AS001973View
2D structure for PGDB_C019190
IC50-=500-1000nM-IKZF3-MGC-803WO2025016359A1PGDB_A031677PGDB_C019190PGDB_AS001973View
2D structure for PGDB_C019181
IC50-=50-100nM-IKZF3-MGC-803WO2025016359A1PGDB_A033786PGDB_C019181PGDB_AS001973View
2D structure for PGDB_C019188
IC50-=100-500nM-IKZF3-MGC-803WO2025016359A1PGDB_A036014PGDB_C019188PGDB_AS001973View
2D structure for PGDB_C019200
IC50-=10-50nM-IKZF3-MGC-803WO2025016359A1PGDB_A036450PGDB_C019200PGDB_AS001973View
2D structure for PGDB_C019204
IC50-=100-500nM-IKZF3-MGC-803WO2025016359A1PGDB_A036870PGDB_C019204PGDB_AS001973View
2D structure for PGDB_C019220
IC50-=100-500nM-IKZF3-MGC-803WO2025016359A1PGDB_A039777PGDB_C019220PGDB_AS001973View
2D structure for PGDB_C019216
IC50-=500-1000nM-IKZF3-MGC-803WO2025016359A1PGDB_A042293PGDB_C019216PGDB_AS001973View
2D structure for PGDB_C019219
IC50-=10-50nM-IKZF3-MGC-803WO2025016359A1PGDB_A044639PGDB_C019219PGDB_AS001973View
2D structure for PGDB_C019191
IC50-=100-500nM-IKZF3-MGC-803WO2025016359A1PGDB_A044817PGDB_C019191PGDB_AS001973View
2D structure for PGDB_C019186
IC50-=500-1000nM-IKZF3-MGC-803WO2025016359A1PGDB_A051913PGDB_C019186PGDB_AS001973View
2D structure for PGDB_C019227
IC50-=5-10nM-IKZF3-MGC-803WO2025016359A1PGDB_A054252PGDB_C019227PGDB_AS001973View