Assay
PGDB_AS002403
System: cell_basedCell line: NCI-H358
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.9045 | nM | - | — | KRAS | - | NCI-H358 | CN121181579A | PGDB_A014069 | PGDB_C011631 | PGDB_AS002403 | View | |
| IC50 | - | = | 4.901 | nM | - | — | KRAS | - | NCI-H358 | CN121181579A | PGDB_A043664 | PGDB_C011587 | PGDB_AS002403 | View | |
| IC50 | - | = | 0.4719 | nM | - | — | KRAS | - | NCI-H358 | CN121181579A | PGDB_A045275 | PGDB_C024627 | PGDB_AS002403 | View | |
| IC50 | - | = | 0.6771 | nM | - | — | KRAS | - | NCI-H358 | CN121181579A | PGDB_A048579 | PGDB_C024673 | PGDB_AS002403 | View | |
| IC50 | - | = | 0.4508 | nM | - | — | KRAS | - | NCI-H358 | CN121181579A | PGDB_A061320 | PGDB_C024605 | PGDB_AS002403 | View | |
| IC50 | - | = | 0.5622 | nM | - | — | KRAS | - | NCI-H358 | CN121181579A | PGDB_A070655 | PGDB_C024617 | PGDB_AS002403 | View |