Summary
AssigneeLinkcure Therapeutics
Filing years2025
Patents1
Compounds115
Activity records231
Patent families1
Targets1
Assay familiesdegradation
Activity metricsDC50, Dmax
Overview

Target distribution and active-compound trend

Target distribution

237 activity records

2 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

0581152025
Activity compounds and values

Activity records

237 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C012089
DC50-=16.6nM-WIZ-HT-1080WO2025256460A1PGDB_A007034PGDB_C012089PGDB_AS000508View
2D structure for PGDB_C012145
DC50-=44.1nM-WIZ-HT-1080WO2025256460A1PGDB_A007446PGDB_C012145PGDB_AS000508View
2D structure for PGDB_C012144
Dmax-=88.5%--WIZ-HT-1080WO2025256460A1PGDB_A007840PGDB_C012144PGDB_AS002062View
2D structure for PGDB_C012093
Dmax-=92.4%--WIZ-HT-1080WO2025256460A1PGDB_A007904PGDB_C012093PGDB_AS002062View
2D structure for PGDB_C012053
Dmax-=88.9%--WIZ-HT-1080WO2025256460A1PGDB_A008226PGDB_C012053PGDB_AS002062View
2D structure for PGDB_C012090
DC50-=10.3nM-WIZ-HT-1080WO2025256460A1PGDB_A008228PGDB_C012090PGDB_AS000508View
2D structure for PGDB_C012106
DC50-=11.9nM-WIZ-HT-1080WO2025256460A1PGDB_A008330PGDB_C012106PGDB_AS000508View
2D structure for PGDB_C012074
Dmax-=90.9%--WIZ-HT-1080WO2025256460A1PGDB_A008761PGDB_C012074PGDB_AS002062View
2D structure for PGDB_C012127
Dmax-=93.5%--WIZ-HT-1080WO2025256460A1PGDB_A008834PGDB_C012127PGDB_AS002062View
2D structure for PGDB_C012067
Dmax-=81.2%--WIZ-HT-1080WO2025256460A1PGDB_A009524PGDB_C012067PGDB_AS002062View
2D structure for PGDB_C012056
Dmax-=92.2%--WIZ-HT-1080WO2025256460A1PGDB_A009686PGDB_C012056PGDB_AS002062View
2D structure for PGDB_C012141
Dmax-=87.7%--WIZ-HT-1080WO2025256460A1PGDB_A010135PGDB_C012141PGDB_AS002062View
2D structure for PGDB_C012077
Dmax-=91.3%--WIZ-HT-1080WO2025256460A1PGDB_A010284PGDB_C012077PGDB_AS002062View
2D structure for PGDB_C012159
Dmax-=89.1%--WIZ-HT-1080WO2025256460A1PGDB_A010328PGDB_C012159PGDB_AS002062View
2D structure for PGDB_C012120
DC50-=23.8nM-WIZ-HT-1080WO2025256460A1PGDB_A010414PGDB_C012120PGDB_AS000508View
2D structure for PGDB_C012110
Dmax-=92%--WIZ-HT-1080WO2025256460A1PGDB_A010751PGDB_C012110PGDB_AS002062View
2D structure for PGDB_C012150
DC50-=7.2nM-WIZ-HT-1080WO2025256460A1PGDB_A010941PGDB_C012150PGDB_AS000508View
2D structure for PGDB_C012116
Dmax-=92.9%--WIZ-HT-1080WO2025256460A1PGDB_A011068PGDB_C012116PGDB_AS002062View
2D structure for PGDB_C012151
DC50-=40.2nM-WIZ-HT-1080WO2025256460A1PGDB_A011136PGDB_C012151PGDB_AS000508View
2D structure for PGDB_C012073
Dmax-=79.5%--WIZ-HT-1080WO2025256460A1PGDB_A011238PGDB_C012073PGDB_AS002062View