Summary
AssigneeWigen Biomedicine Technology Shanghai
Filing years2025
Patents1
Compounds333
Activity records456
Patent families1
Targets1
Assay familiesdegradation, viability
Activity metricsEC50, IC50
Overview

Target distribution and active-compound trend

Target distribution

524 activity records

2 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

01673332025
Activity compounds and values

Activity records

524 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C020732
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A007029PGDB_C020732PGDB_AS001676View
2D structure for PGDB_C020503
IC50-=<= 0.5nM-GSPT1-HEK293TWO2025162410A1PGDB_A007269PGDB_C020503PGDB_AS002143View
2D structure for PGDB_C020605
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A007328PGDB_C020605PGDB_AS001676View
2D structure for PGDB_C020481
IC50-=<= 0.5nM-GSPT1-HEK293TWO2025162410A1PGDB_A007505PGDB_C020481PGDB_AS002143View
2D structure for PGDB_C020499
IC50-=<= 0.5nM-GSPT1-HEK293TWO2025162410A1PGDB_A007633PGDB_C020499PGDB_AS002143View
2D structure for PGDB_C020721
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A007733PGDB_C020721PGDB_AS001676View
2D structure for PGDB_C020682
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A007779PGDB_C020682PGDB_AS001676View
2D structure for PGDB_C020530
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A007803PGDB_C020530PGDB_AS001676View
2D structure for PGDB_C020684
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A007804PGDB_C020684PGDB_AS001676View
2D structure for PGDB_C020538
IC50-=0.5-5nM-GSPT1-HCC1569WO2025162410A1PGDB_A007831PGDB_C020538PGDB_AS001676View
2D structure for PGDB_C020693
IC50-=0.5-5nM-GSPT1-HCC1569WO2025162410A1PGDB_A008034PGDB_C020693PGDB_AS001676View
2D structure for PGDB_C020741
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A008073PGDB_C020741PGDB_AS001676View
2D structure for PGDB_C020554
IC50-=0.5-5nM-GSPT1-HCC1569WO2025162410A1PGDB_A008292PGDB_C020554PGDB_AS001676View
2D structure for PGDB_C020771
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A008331PGDB_C020771PGDB_AS001676View
2D structure for PGDB_C020521
IC50-=0.5-5nM-GSPT1-HCC1569WO2025162410A1PGDB_A008445PGDB_C020521PGDB_AS001676View
2D structure for PGDB_C020477
EC50-=<= 0.5nM-GSPT1--WO2025162410A1PGDB_A008456PGDB_C020477PGDB_AS002258View
2D structure for PGDB_C020585
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A008788PGDB_C020585PGDB_AS001676View
2D structure for PGDB_C020665
IC50-<=0.5nM-GSPT1-HCC1569WO2025162410A1PGDB_A008887PGDB_C020665PGDB_AS001676View
2D structure for PGDB_C020501
Selectivity index-=10-100fold----WO2025162410A1PGDB_A009134PGDB_C020501PGDB_AS000299View
2D structure for PGDB_C020478
EC50-=<= 0.5nM-GSPT1--WO2025162410A1PGDB_A009253PGDB_C020478PGDB_AS002258View