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Compound
PGDB_C002229
5 activity records1 related patents
2D structure
O=C1CCC(N2C(=O)c3cccc(NCc4cccc(C(=O)NC5CCC(c6nc7ccccc7o6)CC5)c4)c3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GI50 | - | = | 0.96 | nM | - | — | GSPT1 | - | Toledo | WO2023237116A1 | PGDB_A014475 | PGDB_C002229 | PGDB_AS002036 | View |
| GI50 | - | < | 100 | nM | - | — | GSPT1 | - | HL-60 | WO2023237116A1 | PGDB_A021947 | PGDB_C002229 | PGDB_AS001555 | View |
| DC50 | - | < | 100 | nM | - | — | GSPT1 | - | HEK293 | WO2023237116A1 | PGDB_A031313 | PGDB_C002229 | PGDB_AS002200 | View |
| GI50 | - | = | 4.07 | nM | - | — | GSPT1 | - | SU-DHL-2 | WO2023237116A1 | PGDB_A036141 | PGDB_C002229 | PGDB_AS000205 | View |
| GI50 | - | = | 1.36 | nM | - | — | GSPT1 | - | NCI-H929 | WO2023237116A1 | PGDB_A038872 | PGDB_C002229 | PGDB_AS000710 | View |