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Compound
PGDB_C007968
4 activity records1 related patents
2D structure
Cc1cccc2nc(COC(=O)NCc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4)sc12Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 30 | % | 10 uM | 6 h | CDK2 | - | HEK293 | WO2025043225 | PGDB_A034617 | PGDB_C007968 | PGDB_AS002435 | View |
| IC50 | - | = | 0.063 | uM | - | — | CRBN | CRBN | - | WO2025043225 | PGDB_A042485 | PGDB_C007968 | PGDB_AS001908 | View |
| IC50 | - | = | 10 | uM | - | — | GSPT1 | - | HEK293 | WO2025043225 | PGDB_A058369 | PGDB_C007968 | PGDB_AS002153 | View |
| IC50 | - | = | 0.067 | uM | - | — | CDK2 | - | HEK293 | WO2025043225 | PGDB_A069499 | PGDB_C007968 | PGDB_AS002528 | View |