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Compound
PGDB_C019869
9 activity records1 related patents
2D structure
CSc1ccccc1C(=O)Nc1nc2nc(C)cc(C)c2s1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000286 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A023821 | PGDB_C019869 | PGDB_AS002126 | View |
| EC50 | - | = | 0.0000536 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A029383 | PGDB_C019869 | PGDB_AS000046 | View |
| EC50 | - | = | 0.0000299 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A032796 | PGDB_C019869 | PGDB_AS002246 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A038770 | PGDB_C019869 | PGDB_AS001009 | View |
| Dmax | - | = | 0.18 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A039038 | PGDB_C019869 | PGDB_AS000856 | View |
| Dmax | - | = | 83.05 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A041485 | PGDB_C019869 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000014 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A067972 | PGDB_C019869 | PGDB_AS001078 | View |
| Dmax | - | = | 23.51 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A071132 | PGDB_C019869 | PGDB_AS001280 | View |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A077100 | PGDB_C019869 | PGDB_AS001381 | View |