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SIMM · NJU
Assay
PGDB_AS000046
System: biochemical
Target: FBXW7
Assay context summary
Assay context
58 activity records
Assay family
biochemical
System
biochemical
Readout
EC50
Target
FBXW7
E3
Not specified
Activity compounds and values
Activity records
58 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
=
0.0000127
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A007442
PGDB_C019915
PGDB_AS000046
View
EC50
-
=
0.0000000032
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A007727
PGDB_C019897
PGDB_AS000046
View
EC50
-
=
0.0000196
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A008208
PGDB_C019880
PGDB_AS000046
View
EC50
-
=
0.0000715
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A008763
PGDB_C019874
PGDB_AS000046
View
EC50
-
=
0.0000000903
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A009207
PGDB_C019917
PGDB_AS000046
View
EC50
-
=
0.0000238
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A009365
PGDB_C019903
PGDB_AS000046
View
EC50
-
=
0.0000000034
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A009689
PGDB_C019907
PGDB_AS000046
View
EC50
-
=
0.0000134
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A009964
PGDB_C019885
PGDB_AS000046
View
EC50
-
=
0.0000014
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A012428
PGDB_C019922
PGDB_AS000046
View
EC50
-
=
0.0000000054
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A014340
PGDB_C019905
PGDB_AS000046
View
EC50
-
=
0.0000221
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A014471
PGDB_C019895
PGDB_AS000046
View
EC50
-
=
0.0000000401
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A016462
PGDB_C019916
PGDB_AS000046
View
EC50
-
=
0.0000186
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A016849
PGDB_C019876
PGDB_AS000046
View
EC50
-
=
0.0000076
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A019640
PGDB_C019886
PGDB_AS000046
View
EC50
-
=
0.0000315
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A020700
PGDB_C019875
PGDB_AS000046
View
EC50
-
=
0.0000174
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A021729
PGDB_C019882
PGDB_AS000046
View
EC50
-
=
0.0000071
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A022838
PGDB_C019910
PGDB_AS000046
View
EC50
-
=
0.0000000412
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A023960
PGDB_C019908
PGDB_AS000046
View
EC50
-
=
0.0000151
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A024961
PGDB_C019901
PGDB_AS000046
View
EC50
-
=
0.0000000082
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A026229
PGDB_C019904
PGDB_AS000046
View