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SIMM · NJU
Assay
PGDB_AS001009
System: biochemical
Target: FBXW7
Assay context summary
Assay context
58 activity records
Assay family
biochemical
System
biochemical
Readout
EC50
Target
FBXW7
E3
Not specified
Technology
luminescence
Activity compounds and values
Activity records
58 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A007624
PGDB_C019896
PGDB_AS001009
View
EC50
-
=
0.0000754
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A008024
PGDB_C019868
PGDB_AS001009
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A008738
PGDB_C019889
PGDB_AS001009
View
EC50
-
=
0.000054
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A012465
PGDB_C019880
PGDB_AS001009
View
EC50
-
=
0.0000442
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A013409
PGDB_C019891
PGDB_AS001009
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A015612
PGDB_C019888
PGDB_AS001009
View
EC50
-
=
0.0000609
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A016735
PGDB_C019911
PGDB_AS001009
View
EC50
-
=
0.0000404
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A017803
PGDB_C019881
PGDB_AS001009
View
EC50
-
=
0.0000544
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A018000
PGDB_C019910
PGDB_AS001009
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A018435
PGDB_C019875
PGDB_AS001009
View
EC50
-
=
0.0000566
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A018497
PGDB_C019898
PGDB_AS001009
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A019690
PGDB_C019918
PGDB_AS001009
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A019724
PGDB_C019870
PGDB_AS001009
View
EC50
-
=
0.0000459
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A020428
PGDB_C019894
PGDB_AS001009
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A020707
PGDB_C021158
PGDB_AS001009
View
EC50
-
=
0.0000414
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A023535
PGDB_C019909
PGDB_AS001009
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A023680
PGDB_C019893
PGDB_AS001009
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A025685
PGDB_C019920
PGDB_AS001009
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A029807
PGDB_C019892
PGDB_AS001009
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A032390
PGDB_C019874
PGDB_AS001009
View