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SIMM · NJU
Assay
PGDB_AS000546
System: biochemical
Target: FBXW7
Assay context summary
Assay context
60 activity records
Assay family
biochemical
System
biochemical
Readout
Dmax
Target
FBXW7
E3
Not specified
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
60 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
0.06
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A010558
PGDB_C019923
PGDB_AS000546
View
Dmax
-
=
0.11
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A011767
PGDB_C019916
PGDB_AS000546
View
Dmax
-
=
1.65
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A012885
PGDB_C019904
PGDB_AS000546
View
Dmax
-
=
-0.2742
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A014245
PGDB_C019870
PGDB_AS000546
View
Dmax
-
=
0.24
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A014342
PGDB_C019886
PGDB_AS000546
View
Dmax
-
=
3
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A016562
PGDB_C019906
PGDB_AS000546
View
Dmax
-
=
2.7
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A019973
PGDB_C019920
PGDB_AS000546
View
Dmax
-
=
-0.2468
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A020011
PGDB_C019912
PGDB_AS000546
View
Dmax
-
=
2.77
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A020650
PGDB_C019880
PGDB_AS000546
View
Dmax
-
=
1.56
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A020666
PGDB_C021158
PGDB_AS000546
View
Dmax
-
=
3.64
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A021801
PGDB_C019891
PGDB_AS000546
View
Dmax
-
=
-0.0757
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A022140
PGDB_C019921
PGDB_AS000546
View
Dmax
-
=
0.32
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A023261
PGDB_C019908
PGDB_AS000546
View
Dmax
-
=
0.86
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A023518
PGDB_C019910
PGDB_AS000546
View
Dmax
-
=
29.69
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A024025
PGDB_C019925
PGDB_AS000546
View
Dmax
-
=
0.65
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A028614
PGDB_C019874
PGDB_AS000546
View
Dmax
-
=
-0.1894
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A031649
PGDB_C019915
PGDB_AS000546
View
Dmax
-
=
4.23
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A031886
PGDB_C019894
PGDB_AS000546
View
Dmax
-
=
-0.4222
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A032722
PGDB_C019914
PGDB_AS000546
View
Dmax
-
=
0.27
%
-
-
FBXW7
-
-
WO2019200310A1
PGDB_A033047
PGDB_C021159
PGDB_AS000546
View