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SIMM · NJU
Assay
PGDB_AS002246
System: biochemical
Target: FBXW7
Assay context summary
Assay context
60 activity records
Assay family
biochemical
System
biochemical
Readout
EC50
Target
FBXW7
E3
Not specified
Activity compounds and values
Activity records
60 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
=
0.0000593
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A009057
PGDB_C019914
PGDB_AS002246
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A010673
PGDB_C019888
PGDB_AS002246
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A013321
PGDB_C019867
PGDB_AS002246
View
EC50
-
=
0.0000432
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A013932
PGDB_C019908
PGDB_AS002246
View
EC50
-
=
0.0000672
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A015231
PGDB_C019879
PGDB_AS002246
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A015845
PGDB_C019920
PGDB_AS002246
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A016188
PGDB_C019917
PGDB_AS002246
View
EC50
-
=
0.0000453
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A017742
PGDB_C019884
PGDB_AS002246
View
EC50
-
=
0.0000567
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A018118
PGDB_C019916
PGDB_AS002246
View
EC50
-
=
0.0000566
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A020187
PGDB_C019913
PGDB_AS002246
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A021925
PGDB_C019887
PGDB_AS002246
View
EC50
-
=
0.0000609
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A022927
PGDB_C019911
PGDB_AS002246
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A025622
PGDB_C021157
PGDB_AS002246
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A026065
PGDB_C019924
PGDB_AS002246
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A027291
PGDB_C019893
PGDB_AS002246
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A029427
PGDB_C019922
PGDB_AS002246
View
EC50
-
=
0.0000729
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A031796
PGDB_C019904
PGDB_AS002246
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A032160
PGDB_C019872
PGDB_AS002246
View
EC50
-
=
0.0000653
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A032529
PGDB_C019889
PGDB_AS002246
View
EC50
-
=
0.0000299
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A032796
PGDB_C019869
PGDB_AS002246
View