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SIMM · NJU
Assay
PGDB_AS002126
System: biochemical
Target: FBXW7
Assay context summary
Assay context
60 activity records
Assay family
biochemical
System
biochemical
Readout
EC50
Target
FBXW7
E3
Not specified
Activity compounds and values
Activity records
60 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
=
0.0000142
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A007266
PGDB_C019882
PGDB_AS002126
View
EC50
-
=
0.0000022
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A007401
PGDB_C021159
PGDB_AS002126
View
EC50
-
=
0.0000000001318
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A008072
PGDB_C019883
PGDB_AS002126
View
EC50
-
=
0.0000000203
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A008602
PGDB_C019887
PGDB_AS002126
View
EC50
-
=
0.0000164
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A009201
PGDB_C019894
PGDB_AS002126
View
EC50
-
=
0.0000241
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A009333
PGDB_C019900
PGDB_AS002126
View
EC50
-
=
0.0000023
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A010864
PGDB_C019919
PGDB_AS002126
View
EC50
-
=
0.0000245
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A012380
PGDB_C019910
PGDB_AS002126
View
EC50
-
=
0.0000116
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A014099
PGDB_C019888
PGDB_AS002126
View
EC50
-
=
0.0000041
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A014225
PGDB_C021158
PGDB_AS002126
View
EC50
-
=
0.0000212
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A014433
PGDB_C019874
PGDB_AS002126
View
EC50
-
=
0.0000202
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A014574
PGDB_C019899
PGDB_AS002126
View
EC50
-
=
0.0001255
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A015960
PGDB_C019908
PGDB_AS002126
View
EC50
-
=
0.0000476
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A016545
PGDB_C019871
PGDB_AS002126
View
EC50
-
=
0.0000286
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A023821
PGDB_C019869
PGDB_AS002126
View
EC50
-
=
0.0000000053
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A024137
PGDB_C019881
PGDB_AS002126
View
EC50
-
=
0.0000212
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A024689
PGDB_C019895
PGDB_AS002126
View
EC50
-
=
0.0000139
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A024740
PGDB_C019915
PGDB_AS002126
View
EC50
-
=
0.000019
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A025061
PGDB_C021157
PGDB_AS002126
View
EC50
-
=
0.0000119
M
-
—
FBXW7
-
-
WO2019200310A1
PGDB_A025792
PGDB_C019920
PGDB_AS002126
View