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COc1ccccc1-c1ccc(N2CCN(C(=O)COc3ccccc3)CC2)nn1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | -0.2742 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A014245 | PGDB_C019870 | PGDB_AS000546 | View | |
| Dmax | - | = | 23.1 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A016587 | PGDB_C019870 | PGDB_AS001280 | View | |
| Dmax | - | = | 0.32 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A017166 | PGDB_C019870 | PGDB_AS000856 | View | |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A019724 | PGDB_C019870 | PGDB_AS001009 | View | |
| EC50 | - | = | 0.000018 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A035290 | PGDB_C019870 | PGDB_AS000046 | View | |
| EC50 | - | = | 0.0000000059 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A059641 | PGDB_C019870 | PGDB_AS002126 | View | |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A060847 | PGDB_C019870 | PGDB_AS002246 | View | |
| EC50 | - | = | 0.0000000881 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A065893 | PGDB_C019870 | PGDB_AS001078 | View | |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A075490 | PGDB_C019870 | PGDB_AS001381 | View |