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Compound
PGDB_C019871
9 activity records1 related patents
2D structure
CCSc1nnc(C2CCN(CC(=O)Nc3cccc4cc(C)ccc34)CC2)n1CCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000476 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A016545 | PGDB_C019871 | PGDB_AS002126 | View |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A023092 | PGDB_C019871 | PGDB_AS001381 | View |
| EC50 | - | = | 0.0000007992 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A023851 | PGDB_C019871 | PGDB_AS001078 | View |
| Dmax | - | = | 0.22 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A057555 | PGDB_C019871 | PGDB_AS000856 | View |
| EC50 | - | = | 0.000018 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A059869 | PGDB_C019871 | PGDB_AS000046 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A064713 | PGDB_C019871 | PGDB_AS001009 | View |
| Dmax | - | = | 0.67 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A067429 | PGDB_C019871 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A070033 | PGDB_C019871 | PGDB_AS002246 | View |
| Dmax | - | = | 22.9 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A071035 | PGDB_C019871 | PGDB_AS001280 | View |