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Compound
PGDB_C019874
9 activity records1 related patents
2D structure
CCc1ccc(-c2cnc(N3CCN(C(=O)c4cccs4)CC3)c3nccn23)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000715 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A008763 | PGDB_C019874 | PGDB_AS000046 | View |
| Dmax | - | = | 1.13 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A011395 | PGDB_C019874 | PGDB_AS000856 | View |
| EC50 | - | = | 0.0000212 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A014433 | PGDB_C019874 | PGDB_AS002126 | View |
| EC50 | - | = | 0.0012 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A016377 | PGDB_C019874 | PGDB_AS001078 | View |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A020074 | PGDB_C019874 | PGDB_AS001381 | View |
| Dmax | - | = | 0.65 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A028614 | PGDB_C019874 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A032390 | PGDB_C019874 | PGDB_AS001009 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A048108 | PGDB_C019874 | PGDB_AS002246 | View |
| Dmax | - | = | 20.66 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A072393 | PGDB_C019874 | PGDB_AS001280 | View |