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O=C(c1ccco1)N1CCN(c2ncc(-c3ccccc3CO)n3ccnc23)CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 0.18 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A027923 | PGDB_C019877 | PGDB_AS000856 | View | |
| EC50 | - | = | 0.000024 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A041713 | PGDB_C019877 | PGDB_AS001078 | View | |
| Dmax | - | = | 18.08 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A047541 | PGDB_C019877 | PGDB_AS001280 | View | |
| Dmax | - | = | 0.83 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A061045 | PGDB_C019877 | PGDB_AS000546 | View | |
| EC50 | - | = | 0.0000203 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A062641 | PGDB_C019877 | PGDB_AS000046 | View | |
| EC50 | - | = | 0.0000002294 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A064204 | PGDB_C019877 | PGDB_AS002126 | View | |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A074356 | PGDB_C019877 | PGDB_AS001009 | View | |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A075068 | PGDB_C019877 | PGDB_AS002246 | View | |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A077184 | PGDB_C019877 | PGDB_AS001381 | View |