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O=C(Nc1ccc2c(c1)OCO2)N1CCC(c2nnc(C3CC3)s2)CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000000575 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A010106 | PGDB_C019878 | PGDB_AS001078 | View | |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A013072 | PGDB_C019878 | PGDB_AS001381 | View | |
| Dmax | - | = | 0.08 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A015192 | PGDB_C019878 | PGDB_AS000856 | View | |
| EC50 | - | = | 0.0000319 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A039727 | PGDB_C019878 | PGDB_AS000046 | View | |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A043843 | PGDB_C019878 | PGDB_AS001009 | View | |
| Dmax | - | = | 0.2 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A048380 | PGDB_C019878 | PGDB_AS000546 | View | |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A064745 | PGDB_C019878 | PGDB_AS002246 | View | |
| EC50 | - | = | 0.0000245 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A069068 | PGDB_C019878 | PGDB_AS002126 | View | |
| Dmax | - | = | 17.46 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A076618 | PGDB_C019878 | PGDB_AS001280 | View |