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Cc1ccc(-c2nnc(N3CCN(C(=O)c4ccco4)CC3)c3ccccc23)cc1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000196 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A008208 | PGDB_C019880 | PGDB_AS000046 | View | |
| EC50 | - | = | 0.000054 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A012465 | PGDB_C019880 | PGDB_AS001009 | View | |
| EC50 | - | = | 0.0000000071 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A013825 | PGDB_C019880 | PGDB_AS001078 | View | |
| Dmax | - | = | 2.77 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A020650 | PGDB_C019880 | PGDB_AS000546 | View | |
| EC50 | - | = | 0.000054 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A028347 | PGDB_C019880 | PGDB_AS001381 | View | |
| EC50 | - | = | 0.000000008 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A032701 | PGDB_C019880 | PGDB_AS002126 | View | |
| EC50 | - | = | 0.000054 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A056090 | PGDB_C019880 | PGDB_AS002246 | View | |
| Dmax | - | = | 16.54 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A056924 | PGDB_C019880 | PGDB_AS001280 | View | |
| Dmax | - | = | 1.77 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A060547 | PGDB_C019880 | PGDB_AS000856 | View |