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Compound
PGDB_C019881
9 activity records1 related patents
2D structure
CCc1ccc(N2CC(C(=O)NCC(C)(C)CNC(=O)C3CC(=O)N(c4ccc(CC)cc4)C3)CC2=O)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000404 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A017803 | PGDB_C019881 | PGDB_AS001009 | View |
| EC50 | - | = | 0.0000000053 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A024137 | PGDB_C019881 | PGDB_AS002126 | View |
| EC50 | - | = | 0.0000000019 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A028279 | PGDB_C019881 | PGDB_AS001078 | View |
| Dmax | - | = | 2.72 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A035352 | PGDB_C019881 | PGDB_AS000856 | View |
| EC50 | - | = | 0.0000404 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A042337 | PGDB_C019881 | PGDB_AS001381 | View |
| Dmax | - | = | 16.53 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A054947 | PGDB_C019881 | PGDB_AS001280 | View |
| Dmax | - | = | 2.4 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A063237 | PGDB_C019881 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000404 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A067795 | PGDB_C019881 | PGDB_AS002246 | View |
| EC50 | - | = | 0.0000071 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A073465 | PGDB_C019881 | PGDB_AS000046 | View |