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Compound
PGDB_C019882
9 activity records1 related patents
2D structure
CCN1C(=O)c2cccc3c(N4CCCC4)ccc(c23)C1=OCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000142 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A007266 | PGDB_C019882 | PGDB_AS002126 | View |
| EC50 | - | = | 0.0000000000502 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A010551 | PGDB_C019882 | PGDB_AS001078 | View |
| Dmax | - | = | 16.33 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A019265 | PGDB_C019882 | PGDB_AS001280 | View |
| EC50 | - | = | 0.0000174 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A021729 | PGDB_C019882 | PGDB_AS000046 | View |
| Dmax | - | = | 0.35 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A033182 | PGDB_C019882 | PGDB_AS000856 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A042935 | PGDB_C019882 | PGDB_AS002246 | View |
| EC50 | - | = | 0.0000653 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A052866 | PGDB_C019882 | PGDB_AS001381 | View |
| Dmax | - | = | 8.96 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A058273 | PGDB_C019882 | PGDB_AS000546 | View |
| EC50 | - | = | 0.0000653 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A059755 | PGDB_C019882 | PGDB_AS001009 | View |