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COc1cc2c(cc1OC)C(COc1ccc([N+](=O)[O-])cc1)N(C(=O)c1ccc3c(c1)OCO3)CC2| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.0000000001318 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A008072 | PGDB_C019883 | PGDB_AS002126 | View | |
| EC50 | - | = | 0.0000000055 | M | - | — | CYCEP | - | - | WO2019200310A1 | PGDB_A027775 | PGDB_C019883 | PGDB_AS001078 | View | |
| Dmax | - | = | 1.58 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A035078 | PGDB_C019883 | PGDB_AS000546 | View | |
| EC50 | - | = | 0.0000498 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A036651 | PGDB_C019883 | PGDB_AS001009 | View | |
| EC50 | - | = | 0.0000498 | M | - | — | CYCEP | - | CyCEP | WO2019200310A1 | PGDB_A036925 | PGDB_C019883 | PGDB_AS001381 | View | |
| Dmax | - | = | 2.58 | % | - | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A046882 | PGDB_C019883 | PGDB_AS000856 | View | |
| Dmax | - | = | 16.04 | % | Concentration context: 65.3E-6 | - | FBXW7 | - | - | WO2019200310A1 | PGDB_A047287 | PGDB_C019883 | PGDB_AS001280 | View | |
| EC50 | - | = | 0.0000498 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A052663 | PGDB_C019883 | PGDB_AS002246 | View | |
| EC50 | - | = | 0.0000092 | M | - | — | FBXW7 | - | - | WO2019200310A1 | PGDB_A062409 | PGDB_C019883 | PGDB_AS000046 | View |